Total synthesis and biological evaluation of (+)- and (-)-Butyl ester of rosmarinic acid.
نویسندگان
چکیده
An efficient method for the synthesis of the natural product (+)-(R)-butyl ester of rosmarinic acid (+)-(R)-1 and its enantiomer ( - )-(S)-1 has been developed by chemical resolution of its phenyl lactic acid precursors 4 with ( - )-menthol. Their antioxidative and anti-tumor activities were evaluated.
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عنوان ژورنال:
- Journal of Asian natural products research
دوره 8 6 شماره
صفحات -
تاریخ انتشار 2006